I-Aspirin esebenzayo ephezulu ye-antipyretic ne-analgesic
Incazelo Yomkhiqizo
I-Aspiriningamuncwa ngokushesha engxenyeni yangaphambili yesisu kanye namathumbu amancane ngemva kokuthatha i-aspirin esilwaneni esisodwa sesisu. Izinkomo nezimvu zimunca kancane, cishe i-70% yezinkomo ziyamuncwa, isikhathi esiphezulu sokuhlushwa kwegazi amahora angu-2 ~ 4, kanti isigamu sokuphila amahora angu-3.7. Izinga lakhe lokubopha amaprotheni e-plasma lalingama-70% ~ 90% kuwo wonke umzimba. Ingangena ubisi, kodwa ukugxila kuphansi kakhulu, kungaphinde kudlule emgodleni we-placenta. i-hydrolyzed kancane ibe yi-salicylic acid ne-acetic acid esiswini, i-plasma, amangqamuzana egazi abomvu kanye nezicubu. Ikakhulukazi kumetabolism yesibindi, ukwakheka kwe-glycine ne-glucuronide junction. Ngenxa yokuntuleka kwe-gluconate transferase, ikati linengxenye ende yokuphila futhi liyazwela kulo mkhiqizo.
Isicelo
Ukuze ekwelapheni imfiva, rheumatism, nerve, imisipha, ubuhlungu bamalunga, ukuvuvukala kwezicubu ezithambile kanye negout ezilwaneni.